What are prohormones?

Prohormones amakhemikhali afana nokwakheka nezakhiwo ku-testosterone ne-19-nortestosterone (nandrolone). Lezi yizandulela zemvelo zamahomoni ezocansi noma ziyakwazi ukuguqulwa zenziwe ama-analogs azo ngendlela efanayo yokuguqula umzimba. I-testosterone iyi-hormone yobulili besilisa; kunikeza umphumela obonakalayo we-anabolic, ukwanda kwesisindo, futhi kuthinta uhlelo lwezinzwa, kuqeda ukukhathala futhi kukhulise ithoni nemodi ejwayelekile.

Kalula nje, lezi yizidakamizwa okuthi uma uziphuzile, ziguqulwe zibe yi-testosterone.

Prohormones bathola ukuthandwa ngokomzimba nangokwakha umzimba. Ngenxa yokusetshenziswa kwezidakamizwa, abagijimi bayakwazi ukufeza umphumela omuhle lapho bethola isisindo. Ukubuyekezwa kubonisa ukuthi ukusetshenziswa okuvamile kwe-designer steroids akubangeli imiphumela emibi. Izinto azinazo izinzuzo zemithi ngaphezu kwezidakamizwa ze-anabolic.

Ama-prohormones noma ama-steroid?

Okwamanje, kunjalo, prohormone engcono kakhulu ayikwazi ukuncintisana nezinhlobo ezisebenza kahle zomjovo we-classic anabolic steroids, kepha lona umsebenzi wesikhathi eside. Kumele kuqashelwe ukuthi manje, ukwandisa umphumela we-anabolic, prohormones zisetshenziswa ngasikhathi sinye ngezindlela eziningi:

  • Amanye amafomu ayisisekelo, imvamisa ama-gel capsules, asetshenziswa ngokudla.
  • Ezinye izinhlobo zempuphu noma amaphilisi azoncelwa ngaphansi kolimi, emlonyeni imizuzu engu-30-60 ngaphambi kokuqeqeshwa.
  • Kusishelwa ngokukhethekile nokugcotshwa ngemuva kokuqeqeshwa ukuhlanza isikhumba ukumunca okungu-transdermal.

Futhi siyakwazi ukuthola inhlanganisela enjalo yamafomu ayisisekelo, izilimi ezingezansi, nama-transdermal, avela kahle kakhulu.

Enye inkinga ukuthi igcinwa kanjani prohormones emzimbeni. Isibindi simi ngendlela yeprohormones ngesithiyo esingaweleki. Ngemuva kwalokho ama-80% -90% we prohormones zikhishwe ngaphandle kokufinyelela kumaseli ahlosiwe wezicubu zemisipha, lapho kuhlelwe khona umsebenzi wazo we-anabolic. Ngakho-ke ukuthola umphumela ongaqhathaniswa nalowo wamathebulethi angu-5 mg we-methandrostenolone noma i-stanozolol (ama-anabolic steroids aneqembu le-17-alpha-methyl, elidlula esibindini bese lingena egazini), kudingeka isilinganiso sama-prohormones ka-100 mg noma ngaphezulu. . Le nkinga ixazululwe ngemuva kokwenza amafomu aguquliwe we prohormone engcono kakhulu, ekwazi ukudlula esibindini futhi itholakale ezicutshini zemisipha yomngcele, kufaka phakathi neqembu le-17-alpha-methyl.

Izici ze-prohormones

Izici ze-prohormones

Abaklami be-steroid, lapho bengeniswa, baguqulwa baba yi-hormone eyinhloko. Kukhona okwemvelo ama-prohormones, i-proinsulin, ne-thyroxine emzimbeni womuntu iguqulwe yaba yi-triiodothyronine. Ochwepheshe nodokotela bathi akukho miphumela emibi yezidakamizwa, futhi umzimba womuntu ubona izinto njengezendalo. Umehluko omkhulu phakathi kwe- prohormone engcono kakhulu futhi i-anabolic steroids elula ukuthi izinto ziguqulwa zibe yifomu elisebenzayo ngokushesha bese ziqala ukusebenza. Ama-steroids asemthethweni zisebenza kangcono kakhulu, kepha kukhona imiphumela engemihle emzimbeni.

Amazinga e-Estrogen ne-testosterone ancipha ngobudala; kungashiwo okufanayo ngama-prohormone. Ucwaningo lomtholampilo lukhombisile ukuthi ama-milligram ama-5 ngosuku anele kwabesifazane ngesikhathi sokunqamuka kokuya esikhathini, futhi noma ama-milligram ayishumi ngosuku awasebenzi kwabesilisa. Ukuqeqeshwa njalo akusizi isimo futhi. Ososayensi baqhubeka nokuhlola izidakamizwa, okwagcina kuholele emphumeleni osebenzayo. Okwabesilisa, a isilinganiso wama-milligram angama-20 ngosuku kwanele ukufeza imiphumela emihle. Ama-prohormones athinta ukukhula kwe-testosterone ne-estrogen. Abesifazane abane-hormone therapy basebenzisa le mithi ngesikhathi sokunqamuka kokuya esikhathini.

Ama-prohormones amahle kakhulu

  • I-4-androstenedione iguqulwa ibe yi-testosterone. Ucwaningo lukhombisa ukuthi izinga lokuguqulwa alidluli ku-6%, okusho ukuthi kuphela amashumi amabili wesengezo aguqulwa abe yi-testosterone. Izinga eliphakeme lokunambitheka, okungukuthi, amathuba okuthuthukisa i-gynecomastia, i-edema, nokunye okuqhamuka uma udla imishanguzo, liphezulu. Inomsebenzi ophezulu we-androgenic.
  • I-4-androstenediol (4-AD) iguqulelwa ku-testosterone. Izinga lokuguqulwa elingu-15.76%. Ayiguqulwa ibe yi-estrogen. Inomsebenzi omncane we-androgenic ngokuqhathaniswa ne-4-androstenedione ngoba ayiguqulwa ibe yi-dihydrotestosterone.
  • I-19-norandrostenedione iguqulelwa ku-nandrolone (retabolil). Umsebenzi we-Anabolic ucishe ufane ne-testosterone. Ayiguquli ibe yi-estrogen, futhi inomsebenzi ophansi we-androgenic.
  • 19-noma i-androstenediol, i prohormone engcono kakhulu, ibuye iguqulwe ibe yi-nandrolone. Izinga lokuguqulwa liphakeme kancane kune-prohormone yangaphambilini.
  • I-1-androstenediol (1-AD) iguqulelwe ku-1-testosterone (I-dihydroboldenone). Inomsebenzi omkhulu we-anabolic ophindwe kasikhombisa nomsebenzi omkhulu we-androgenic ophindwe kabili uma kuqhathaniswa ne-testosterone. Cishe iguqulwe ngokuphelele ifomu elisebenzayo lapho udlula esibindini. Akunamakha (ayiguquli ibe yi-estrogen).
  • I-1,4-androstadienedione (1,4 AD) iguqulelwa ku-boldenone. Ukutholakala okuphezulu komlomo. Izinga eliphansi lokunambitheka kwe-estrogen (ngama-50% ngaphansi uma kuqhathaniswa ne-testosterone). Umsebenzi ophansi we-androgenic.
  • I-1-testosterone (1-T) iyafana ne-testosterone. Inokutholakala kokutholakala ngomlomo okuphindwe kane uma kuqhathaniswa ne-testosterone futhi ayiguquli ibe yi-estrogen. Akuyona i-prohormone.

Ungakwazi thenga ama-prohormones e-UK. Kumele uthenge le mithi kubathengisi abathembekile abathengisa kuphela imikhiqizo esezingeni.

Ama-prohormones ekwakheni umzimba

Ama-prohormones ekwakheni umzimba

Eminyakeni engamashumi amabili edlule, prohormone engcono kakhulu isetshenziswe ngenkuthalo ngabasubathi ekwakheni umzimba, ekuphakamiseni amandla, nakweminye imidlalo yezemidlalo ukukhulisa isisindo namandla. Ekuqaleni, inzuzo enkulu yama-prohormones kwakungokwabo zomthetho status njengoba bengeyona eye-anabolic ngokusemthethweni i-steroids. Noma kunjalo, ndoday ama-prohormone zifakwe kuhlu kanye ne-steroids eminyakeni yamuva, futhi ukusakazwa kwazo kunqunyelwe.

Umjaho oqhubekayo womkhiqizi kanye nokulawulwa kukahulumeni kuholela kuma-prohormone avela emakethe angadluli noma yiziphi izivivinyo zokwelashwa. Lezi Izithako kuvame ukuba nokubi kakhulu okuqhamuka uma udla imishanguzo ezinzima kakhulu kune-steroids yakudala. Kumele kuqashelwe ukuthi prohormones banesimo sesengezo sokudla, okusho ukuthi ukulawulwa kwekhwalithi yale mikhiqizo kuncane kakhulu kunalokho kwemithi yokwelapha.


Ama-Prohormones angena ajule kwezemidlalo, asuse ama-anabolic steroids akudala. Kunezinkinga eziningana lapha, kepha futhi kunezinzuzo ezithile ezicacile. Izinkinga zilele ngaphezulu ngenkathi kushintshwa idlanzana lamaphilisi e-methandrostenolone nganoma iyiphi inhlanganisela yama-prohormones akunakwenzeka. Kepha isikhathi se-methane noma i-stanozolol sesidlulile, zinqunywa ngokulawulwa kwe-doping amasonto ambalwa ngemuva kokusetshenziswa, ngakho-ke ubungozi bokubanjwa ekulawuleni okungaphandle komncintiswano bukhulu kakhulu.

Kukholakala ukuthi prohormones ayinabuthi kangako futhi awenziwanga amanga. Ngasikhathi sinye, ama-anabolic steroids ajwayelekile ayenziwa ngomgunyathi, futhi manje awusakwazi ngisho nokwethemba amalebula namaphakheji aqinisekisiwe. Ucwaningo luye lwabonisa ukuthi isikhathi sokususwa kwama-prohormones sifushane kakhulu kunaleso se-anabolic steroids ejwayelekile. Ama-Androstenediols awatholakali noma yini ngemuva kwezinsuku ezimbalwa uma iphrofayli ye-steroid ingacindezelwa ngenxa yokusebenzisa ngokweqile ama-anabolic steroids esikhathi esedlule.