SARMS and Ostarine

Umhlahlandlela Ophelele Mayelana Ne-SARMS ne-Ostarine


Noma ngabe umusha ekwakheni umzimba noma uke waba kulo mdlalo isikhashana, ukubonile ukuvuselelwa kokukhetha androgen receptor ama-modulators (ama-SARM). Ngokushesha ziba enye indlela ethandwayo kuma-steroids.

Kepha ayini ama-SARM, ncamashi? Hlobo luni lwemiphumela abangayinikeza? Ngabe zisemthethweni? Ingabe ikhona imiphumela emibi yokuyithatha?

Uma ulandela imihlahlandlela yesilinganiso, ama-SAR afana ne-Ostarine azokusiza ukuthi uthole amandla amangalisayo, ugqoke imisipha, bese uyigcina ngemuva kwalokho. Futhi ngokumangazayo, ungakufeza konke lokhu ngaphandle kwemiphumela emibi evame ukuhambisana nokusetshenziswa kwe-steroid.

Qhubeka ufundele umhlahlandlela wama-SARM — funda ukuthi ziyini, zisebenza kanjani, zithathe ini, nokuthi ungaqala kanjani uhambo lwakho olusha lokwakha umzimba nama-SARM.

Yini ama-SARM?

Ama-modulators akhethiwe we-androgen receptor athulwe kwifayela le- Ama-1940 nguLigand Pharmaceuticals. Zethulwe okokuqala njengokwelashwa komdlavuza, i-osteoporosis, nezinye izifo. Ngemuva kwalokho, babaziwa ngokuthi "ama-SARM steroidal."

Akuzange kuthathe isikhathi eside ukuthi abacwaningi bathole ukuthi “ama-SARMs steroidal” abe nemiphumela engemihle eminingi. Iziguli bezizothola imisipha ngokushesha — kuze kufike kumakhilogremu angama-30 ezinyangeni ezimbalwa nje — kodwa imiphumela emibi eyenze odokotela bakungabaza ukuphepha kwezithasiselo.

I-Steroid nalawa ma-SARM angama-steroidal angadala imiphumela emibi efana ne-gynecomastia, i-libido ephansi, ukulimala kwesibindi, nesifo senhliziyo. AbakwaDokotela abakwazanga ukuqhubeka nokubanika ngendlela yabo yamanje, ngakho-ke bakhohlwa amashumi eminyaka.

Ngama-1990s, izinkampani zaqala ukuzama "ama-SARM angenayo i-steroidal," okuyilokho manje esikubiza ngamaSARM kuphela. Ukwakheka kwamakhemikhali kwalezi zidakamizwa ezimangazayo kusekelwe emaprotheni, ngakho-ke kunikeza izinzuzo cishe ezingekho nemiphumela engemihle.

Zisebenza Kanjani?

Ngaphandle kwemiphumela emibi, abantu abaningi babuza ukusebenza kwamaSARM. Kepha imfihlo yabo iqukethe indlela yabo yokwenza ekhomba ngokukhetha i-androgen receptors. Zisebenza ngokuzibophezela kuma-receptors we-skeletal muscle androgen ngenkathi zigwema ama-receptors ku-prostate nakwezinye izitho.

Ama-SAR asiza imisipha yakho ukuba ikhule, ngaphandle kwemiphumela emibi ejwayelekile ye-steroids, efana ne-prostate ekhulisiwe.

AmaSARM vs Steroids

I-Anabolic steroids (noma "i-steroids" kuphela) isigaba se-testosterone kanye ne-non-testosterone derivatives. Zikhuthaza ukukhula kwemisipha kubantu. Ososayensi baseJalimane bazithuthukisa ngawo-1930, bezama ukuthola onqenqemeni lwama-Olimpiki.

Ukusetshenziswa kwe-steroid akuzange kudume phakathi kwabakhi bomzimba kuze kube maphakathi no-kuya ngasekupheleni kwawo-1950.

Kunezinhlobo eziningana ze-steroids nama-SARM. Yonke inemiphumela efanayo, kepha indlela esebenza ngayo iyahluka. Ama-steroids amaningi azobopha kukho konke ukwamukelwa kwe-androgen, kepha ama-SARM abopha kuphela kwabambalwa abakhethiwe.

Lo mehluko ungabonakala umncane, kepha ngushintsho lomdlalo kubasubathi abangakwazi ukusingatha imiphumela emibi ye-steroids. Ama-SAR ngokuvamile ane-1-5% kuphela yemiphumela emibi engahle ihlangatshezwe ngabasubathi kuma-steroids — kepha angama-80-90% asebenza njengokusetshenziswa kwe-steroid.

AmaSARM vs Prohormones

Ama-Prohormones awahlukile kakhulu kune-steroids. Njengoba ama-steroids enziwa engekho emthethweni, umthetho ucacisa uhlobo oluthile lwamakhemikhali. Esibonelweni, lapho i-US ithengisa ngokungemthetho i-testosterone, bachaza i-molecule i-Androst-4-en-17β-ol-3-one.

Lo mkhuba uvumela izinkampani ezithaka imithi ukuthi zilungise i-molecule ngokungeza i-athomu elilodwa lapho zingakwazi khona. A prohormone ethandwayo unefomula yamakhemikhali kanye ne -ost-4-en-3,17-dione. Le fomula ihluke kancane kune-testosterone eshiwo ngenhla. Uma ufaka i-prohormone, isibindi sakho siyiguqula sibe yi-hormone efana ne-testosterone. Kanjalo nje, uthathe i-steroid.

Kuzwakala kuyindlela elula yokuzungeza umthetho, kepha lezi zithasiselo zeprohormone zivame ukuba nobuthi kune-steroids. Ingozi isekuthini umsebenzi wesibindi sakho okufanele uwenze ukuzicubungula.

Ngakolunye uhlangothi, amaSARM awanayo le nkinga yobuthi. Zitholakala nge-bio, okusho ukuthi zilula ukucubungula isibindi sakho. Ziphephe, yingakho zisatholakala kabanzi kubakhi bomzimba namuhla.

Ziyini Izinzuzo Zokusebenzisa Ama-SARM Ngaphezulu Kwe-Steroids?

Sesivele sixoxile ngokuthi amaSARM aphephe kangakanani kune-steroids futhi anemiphumela engemihle embalwa, kepha kukhona ezinye izinto ezinhle okufanele uzicabangele.

Ezinye izinzuzo Ukuthatha ama-SAR kuma-steroids kufaka:

  • Azinabo ubuthi futhi azibangeli ukulimala kwesibindi.
  • Zandisa ukwanda kwamathambo.
  • Abavale umkhiqizo wakho we-testosterone wemvelo phansi.
  • Bakha imisipha emincane, eminyene.
  • Ululama ngokushesha lapho ubathatha.
  • Bathuthukisa amandla
  • Bangakwazi ukwelapha amalunga nemisipha.

Kungazwakala kukuhle kakhulu ukuthi kunganemba. Noma kunjalo, ungathola amandla amakhulu, ululame ngokushesha kunanini ngaphambili, futhi ube namathambo aphilile, aqine ngaphandle kokuthola imiphumela emibi. Ngabe lokhu kuzwakala njengesivumelwano esimnandi kuwe?

Yini i-Ostarine?

Ostarine ingenye yama-SARM athandwa kakhulu. Yakhiwa yinkampani eyenza imithi eyizigidigidi zamarandi ebizwa ngeMerck ukumisa nokuhlehlisa ukonakala kwemisipha namathambo.

Okwamanje ihlolwa okusha. Abaphenyi banethemba lokuthi i-Ostarine ingasiza iziguli ezinomdlavuza ezihlushwa imisipha namathambo.

Okwamanje, abakhi bomzimba emhlabeni wonke bathenga i-Ostarine futhi bayisebenzisela ukwenza ngcono ukusebenza kwabo ngokomzimba ngezakhiwo zayo ze-anabolic.

I-Ostarine ayivunyelwe yi- I-World Anti-Doping Agency (WADA) ngoba empeleni isebenza ukuthuthukisa ukuzuza kwemisipha nokusebenza, inika abagijimi abathatha amaSARM inzuzo engafanele.

Ongakulindela

Lapho uthatha i-Ostarine, qiniseka ukuthi ikhiqiza imiphumela emihle ngenkathi iyisengezo esimnene kakhulu. Yilokhu okwenza kube yi-SARM ethandwa kakhulu emakethe.

Njengoba i-Ostarine ingacindezeli, akudingeki ukhathazeke ngokukhishwa kwemali. Noma kunjalo, gcina i-PCT yakho isesandleni uma kungenzeka ukuthi ungehlisi amazinga wakho we-hormone abuyele kokujwayelekile.

I-Ostarine inedumela lokuba nemiphumela engemihle kangako, ikhiqize ukuzuza okuncane, futhi ibambelele emisipheni ngesikhathi sokushoda okukhulu kwekhalori. Kuyinhlanganisela eguquguqukayo enhle kakhulu ekuzuzeni imisipha nokusika amafutha, kuya ngezinhloso zakho nokuthi uwasebenzisa kanjani.

Uma ufuna ukuzuza imisipha, lindela ukuzuza phakathi kwamakhilogremu amane kuya kwayishumi ngaphandle kokuthola amafutha kumjikelezo ojwayelekile wamaviki awu-12.

Uma ufuna ukulahlekelwa ngamafutha, ungasebenzisa i-Ostarine bese uya kokushodayo okukhulu kwekhalori lama-calories ayi-500-1000, ngenkathi ugcina imisipha yakho oyitholile. Futhi kuzokwenyusa ukuzuza kwakho kwamandla nokuqina kwezicubu ezithambile, njengamathambo nemisipha — konke lokhu ngenkathi kukhulisa isikhathi sakho sokululama.

Izinkinga ze-Ostarine

Futhi, imiphumela emibi ye-Ostarine imbalwa futhi iphakathi kakhulu, khumbula ukuthi wonke umuntu uphendula kuma-supplements ngokuhlukile.

Uma ulandela imihlahlandlela enconywayo yokulinganisa, ungahle uhambe kahle. Kodwa-ke, uma umthamo uphakeme kakhulu kunalokho okunconyiwe, ungahle ube nemiphumela emibi efana nokujuluka okubandayo nobuthakathaka.

Yiziphi izilinganiso ezinhle kakhulu ze-SARM?

Ngenkathi ama-SARM e-UK ephephe ngokuqhathaniswa, kufanele ube nengqondo futhi uhlakaniphe ngokuthi uwasebenzisa kanjani-njengoba nje ungenza nganoma yisiphi esinye isidakamizwa noma ikhompiyutha.

Hlola ibhodlela ukuthola umthamo onconyiwe futhi ngaso sonke isikhathi qala ekugcineni okuphansi kwalokho okunconywayo. Lelisu likunikeza indawo yokukhula. Uma uqala phezulu, uzishiya ungenandawo ongathuthukela kuyo.

Emithamo ephansi, ungaqeda isidingo sanoma iyiphi i-PCT. Yiba nje uhlakaniphile ngomjikelezo wakho wama-SARM futhi umangale ngezinzuzo ozozithola lapho uzithatha kahle.

Uyithenga kuphi i-Ostarine?

Kufanele njalo uthenge ama-SAR kusuka kumkhiqizi onedumela elihle. Naka ukuthi imikhiqizo itholakala kuphi nokuthi iqinisekiswe ilebhu ngumuntu wesithathu. Inkampani kufanele ikwazi ukufakazela i- ikhwalithi yezithako zabo.

Ngenxa yenkuthalo yakho efanele lapho uthenga ezungeze i-Ostarine e-UK, njengoba ungakhubeka ezinkampanini ezidayisa ama-prohormone bese uzidlulisa njengama-SARM. Benza lokhu ngoba ama-prohormones ayevinjelwe e-2014 futhi izinkampani eziningi zizama ukuqeda uhlu lwazo ngokusho ukuthi zithengisa ama-SARM.

Isisho esithi “kuhle kakhulu ukuthi ungaba yiqiniso” naso silungile uma uthenga ama-SARM. Uma amanani aphansi ngokungakholeki, kungenzeka ubheke ama-SARM angamanga. Lindela ukukhokha cishe u- $ 50 ngokunikezwa kwe-Ostarine kwenyanga eyodwa; ngakho-ke, umjikelezo wamasonto angu-12 onconyiwe uzobiza cishe ama- $ 150.

Zama ama-SARM ngokwakho

Ama-SARM aseseqoqo elisha lamakhemikhali asaqhubeka nokuhlolwa. Ucwaningo olujabulisayo luveza ukuthi zisebenza ngempumelelo emangalisayo ekusizeni abasebenzisi abanentshisekelo ukuthi bathole imisipha, balahlekelwe ngamafutha, futhi bandise amandla ngaphandle kwemiphumela emibi ehambisana ne-steroids.

Sekukonke, amaSARM ayisethi yamakhompiyutha entsha okwamanje eyohlolwa. Yiluphi ucwaningo esinalo olusikisela ukuthi zisebenza ngempumelelo emangalisayo ekusizeni abasebenzisi ukuthi bafake imisipha, balahlekelwe ngamafutha, futhi bathole amandla — konke lokhu kungenxa yemiphumela emibi i-steroids evame ukuletha.

Sithengisa ama-SARM aphezulu nezengezo eziphephile, ezisebenzayo nezisemthethweni. Zenziwe e-UK ziye emazingeni aphezulu kakhulu, zisebenzisa izithako zebanga lemithi. Okwethu I-Reflex Labs Ostarine i-rounder yonke engasetshenziswa yodwa noma isitaki.

Bheka uhlu lwethu olunzulu lwezithasiselo futhi Xhumana nathi uma singakusiza unqume ukuthi yikuphi okulungele wena!